#158380

MZP55 small molecule (tool compound)

Cat. #158380

MZP55 small molecule (tool compound)

Cat. #: 158380

Availability: Please enquire for quantities and pricing

This fee is applicable only for non-profit organisations. If you are a for-profit organisation or a researcher working on commercially-sponsored academic research, you will need to contact our licensing team for a commercial use license.

Contributor

Inventor: Alessio Ciulli

Institute: University of Dundee

Tool Details
Handling
Target Details
References

Tool Details

*FOR RESEARCH USE ONLY

  • Tool name: MZP55 small molecule (tool compound)
  • Molecular formula: C57H70ClN7O10S
  • Description: MZP-55 is a selective degrader of BRD3/4 based on PROTAC technology
  • Molecular weight: 1080.72
  • Solubility: DMSO

Handling

  • Purity: 1080.72 g/mol
  • Shipping conditions: Dry Ice

Target Details

  • Ic50: Kd: 8 nM (Brd4BD2)

References

  • Chan et al. 2018. J Med Chem. 61(2):504-513. PMID: 28595007.