Cat. #153191
CDK inhibitor BS-194 Small Molecule (Tool Compound)
Cat. #: 153191
Sub-type: Inhibitor
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Contributor
Inventor: Simak Ali
Institute: Imperial College London
Tool Details
*FOR RESEARCH USE ONLY
- Tool name: CDK inhibitor BS-194 Small Molecule (Tool Compound)
- Molecular formula: C20H27N5O3
- Tool sub type: Inhibitor
- Description: BS-194 is a selective and potent CDK inhibitor, which inhibits CDK2, CDK1, CDK5, CDK7, and CDK9.
- Purpose: Inhibitor
- Selectivity: CDK1, CDK2, CDK7, and CDK9
- Iupac: (2S,3S)-3-(7-(benzylamino)-3- isopropylpyrazolo[1,5-a]pyrimidin-5- ylamino)butane-1,2,4-triol
- Molecular weight: 385.5
Handling
- Purity: 385.5 g/mol
- Storage conditions: Ambient
- Shipping conditions: Dry Ice
Target Details
- Ic50: CDK2, CDK1, CDK5, CDK7, and CDK9 (IC50=3, 30, 30, 250, and 90 nmol/L, respectively)
Related Tools
- Related tools: CDK7 inhibitor BS-181 Small Molecule (Tool Compound)
References
- J. Med. Chem. 2010, 53, 85088522
